Lukáš Tenora

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Latest publications

Inhibition of microglial glutaminase alleviates chronic stress-induced neurobehavioral and cognitive deficits

M. Huang Y. Li A. Thomas A. Sharma W. Liyanage T. Tichý L. Tenora Y. Su J. Ha N. Hin M. Obayashi P. Majer R. M. Kannan T. Tsukamoto G. Ursini R. Rais B. S. Slusher X. Zhu

Neurotherapeutics 22 (6): e00759 (2025)

Renaissance of 6-Diazo-5-oxo-ʟ-norleucine (DON): Prodrug Strategy as a Promising Tool Leading to Potential Anticancer Drug

L. Tenora

Chemické listy 119 (5): 274−286 (2025)

Discovery of Orally Available Prodrugs of Itaconate and Derivatives

C. B. Lee I. Šnajdr L. Tenora J. Alt S. Gori M. Krečmerová R. M. Maragakis J. Paule S. Tiwari J. Iyer R. Talwar L. Garza P. Majer B. S. Slusher R. Rais

Journal of Medicinal Chemistry 68 (3): 3433–3444 (2025)

Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-L-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery

K. Novotná L. Tenora E. Prchalová J. Paule J. Alt V. Veeravalli J. Lam Y. Wu I. Šnajdr S. Gori V. S. Mettu T. Tsukamoto P. Majer B. S. Slusher R. Rais

Journal of Medicinal Chemistry 66 (22): 15493–15510 (2023)