Kateřina Tenorová

All publications

Latest publications

Therapeutic resurgence of 6-diazo-5-oxo-L-norleucine (DON) through tissue-targeted prodrugs

K. Novotná L. Tenora B. S. Slusher R. Rais

Advances in Pharmacology, in press, Academic Press (2024)

Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-L-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery

K. Novotná L. Tenora E. Prchalová J. Paule J. Alt V. Veeravalli J. Lam Y. Wu I. Šnajdr S. Gori V. S. Mettu T. Tsukamoto P. Majer B. S. Slusher R. Rais

Journal of Medicinal Chemistry 66 (22): 15493–15510 (2023)

Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a]pyrimidin-3-amine scaffold

K. Novotná A. G. Thomas O. Štěpánek B. Murphy N. Hin J. Skácel L. Mueller L. Tenora A. Pal J. Alt J. Wu J. Paule R. Rais B. S. Slusher T. Tsukamoto

European Journal of Medicinal Chemistry 259: 115674 (2023)

Tumor-Targeted Delivery of 6-Diazo-5-oxo-L-norleucine (DON) Using Substituted Acetylated Lysine Prodrugs

L. Tenora J. Alt R. P. Dash A. J. Gadiano K. Novotná V. Veeravalli J. Lam Q. R. Kirkpatrick K. M. Lemberg P. Majer R. Rais B. S. Slusher

Journal of Medicinal Chemistry 62 (7): 3524-3538 (2019)