Latest publications

Extensive targeting of chemical space at the prime side of ketoamide inhibitors of rhomboid proteases by branched substituents empowers their selectivity and potency
European Journal of Medicinal Chemistry 275: 116606 (2024)
Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-L-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery
Journal of Medicinal Chemistry 66 (22): 15493–15510 (2023)
Comprehensive Mechanistic View of the Hydrolysis of Oxadiazole-Based Inhibitors by Histone Deacetylase 6 (HDAC6)
ACS Chemical Biology 18 (7): 1594–1610 (2023)